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Cerebrolysin

Well Studied

Neuropeptide Preparation | Neurological Recovery

Dose 10-50mL depending on indication (stroke/TBI higher doses)
Frequency Once daily for acute conditions; 5 days weekly for chronic conditions
Cycle 7-30 days depending on condition (stroke/TBI 10-30 days, dementia 4 weeks)
Storage Room temperature ≤25°C, protected from light in original carton - never freeze

Community Research

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Standardized neuropeptide preparation containing bioactive peptides and amino acids exhibiting neurotrophic and neuroprotective properties for stroke recovery, traumatic brain injury, and cognitive enhancement. Used clinically in 50+ countries.

Mechanism of Action

IV/IM administration provides optimal bioavailability and brain penetration of neuropeptides and neurotrophic factors.

Key Benefits

  • Direct brain delivery
  • Standardized dosing
  • Extensive clinical evidence
  • Ready-to-use formulation
  • Used clinically in 50+ countries
Molecular Weight
Variable
Chain Length
Multiple peptides
Type
Purified porcine brain proteins
Amino Acid Sequence
Bioactive peptide mixture

Complex or non-standard sequence format

Cognitive

  • Alzheimer's Disease

    Meta-analyses show modest cognitive improvements, though clinical significance remains debated.

  • Vascular Dementia

    Multiple RCTs demonstrate significant ADAS-cog and CIBIC+ improvements.

  • Post-Stroke Cognitive Recovery

    Large meta-analysis shows significant NIHSS improvements; other studies found no functional benefit.

Neuroprotection

  • Acute Stroke

    Largest meta-analysis (1,879 patients) shows NIHSS benefits; independent analysis found no mRS improvement.

  • Traumatic Brain Injury

    Multiple trials including CAPTAIN series confirm GCS/GOS improvements.

  • Subarachnoid Hemorrhage

    Pilot trial shows promising 6-month outcomes; requires larger confirmatory studies.

Recovery

  • Motor Function Recovery

    Some studies show enhanced recovery; results vary significantly between trials.

  • Neurological Function

    Early administration within 72 hours shows better outcomes than delayed treatment.

Primary administration route with well-established protocols for direct brain delivery via IV/IM.

GoalDoseFrequencyRoute
Small Volume IVUp to 10mLOnce dailyUndiluted IV slow push over 3 minutes
IntramuscularUp to 5mLOnce dailyUndiluted IM injection over 3 minutes
Acute Stroke20-50mLOnce daily for 10-21 daysIV infusion (diluted to 100mL minimum)
Traumatic Brain Injury20-50mLOnce daily for 7-30 daysIV infusion (diluted to 100mL minimum)
Alzheimer's Disease10-30mL5 days weekly for 4 weeksIV injection/infusion (2-4 cycles yearly)
Vascular Dementia10-30mL5 days weekly for 4 weeksIV injection/infusion (2-4 cycles yearly)

Reconstitution Instructions

Materials Needed:
  • Cerebrolysin ampoules (5, 10, or 20 mL)
  • Saline, Ringer solution, or 5% glucose (minimum 100 mL for infusion)
  • Disposable one-way IV infusion sets and cannulas
  • Sterile syringes and alcohol swabs
  1. 1 Break ampoule and extract Cerebrolysin immediately before use
  2. 2 For direct injection: Up to 10 mL IV undiluted (slow 3 minutes) or 5 mL IM
  3. 3 For infusion: Dilute 10-50 mL to minimum 100 mL with compatible solution
  4. 4 Start infusion immediately after dilution—infuse within 15 minutes
  5. 5 Flush IV catheter with sodium chloride before and after administration
  6. 6 Use disposable one-way infusion sets; discard after use
Piracetam

Safe combination with no significant interactions; both support cognitive function.

compatible
Donepezil

No interactions reported; may have synergistic cognitive effects in Alzheimer's treatment.

compatible
SSRIs

Potential additive neurotropic effects; monitor for enhanced antidepressant effects.

monitor
Tricyclic Antidepressants

May have additive neurological effects; requires careful monitoring.

monitor
Amino Acid Solutions

Contraindicated per prescribing information; do not mix in same infusion.

avoid
Cardiovascular Medications

Should not be mixed in same IV infusion per official guidelines.

avoid
Vitamin Solutions

Compatibility issues; do not mix in same IV infusion.

avoid
Noopept

Both enhance neurotrophic factors; potential additive effects—start with lower doses.

monitor
Week 1-2

Initial neuroprotective effects; possible mild side effects (dizziness, agitation)

Week 2-4

Neurological improvements become apparent; cognitive function may begin to improve

Week 4-8

Continued recovery; motor function improvements in stroke/TBI patients

Week 8-12

Sustained benefits; cognitive enhancement plateaus in chronic conditions

Common Side Effects

  • Generally well tolerated
  • Possible mild dizziness or agitation in early treatment

Stop Signs - Discontinue if:

  • Severe allergic reactions (anaphylaxis, severe rash)
  • New onset seizure activity
  • Significant cardiovascular events during administration
  • Severe renal dysfunction or worsening kidney function

Contraindications

  • Epilepsy
  • Severe renal insufficiency
  • History of severe allergic reactions to porcine products

Good Signs

  • Clear amber solution from reputable source
  • Room temperature storage ≤25°C
  • Protected from light in original carton
  • Authorized EVER Pharma distributor

Warning Signs

  • Some published studies have been retracted due to research misconduct; rely on independent meta-analyses

Bad Signs

  • Frozen product or improper storage—never freeze
  • Mixing with incompatible solutions (amino acids, vitamins, cardiovascular medications)
  • CAPTAIN II Trial - Traumatic Brain Injury
    (2020)

    Randomized controlled trial demonstrating efficacy and safety in moderate-severe TBI with improved GCS and GOS scores.

  • Nine-Trial Stroke Meta-Analysis - Positive Results
    (2017)

    Largest positive meta-analysis showing significant neurological improvements in 1,879 stroke patients with NNT=7.7.

  • Conflicting Stroke Meta-Analysis - Neutral Results
    (2017)

    Independent meta-analysis of 1,779 patients found no significant benefits in functional outcomes (mRS/BI).

  • TBI Systematic Review - Positive Outcomes
    (2023)

    Analysis of 8,749 TBI patients across 10 studies confirms statistically significant GCS/GOS improvements.

Disclaimer

This information is for educational and research purposes only. Consult a healthcare professional before use.